BDBM50306236 2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-hydroxy-4-(pyridin-2-yl)piperidine-1-carbonyl)-1H-pyrazol-4-yl)acetamide::CHEMBL596166

SMILES NC(=O)Cc1c(nn(c1-c1ccc(Cl)cc1)-c1ccccc1Cl)C(=O)N1CCC(O)(CC1)c1ccccn1

InChI Key InChIKey=LVEYNBFOVLRQTM-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50306236   

TargetCannabinoid receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50306236(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-hydr...)
Affinity DataIC50:  3.60nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940-induced GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50306236(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-hydr...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50306236(2-(1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(4-hydr...)
Affinity DataIC50:  2nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in CHO-K1 cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed